SML1061-25MG Display Image

PF-04856264

Code: SML1061-25MG D2-231

Biochem/physiol Actions

PF-04856264 is a potent, selective inhibitor of the human Nav1.7 voltage gated sodium channel (IC50 = 28 nM). PF-04856264 blocks mouse Nav1...


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£421.00 25MG
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Biochem/physiol Actions

PF-04856264 is a potent, selective inhibitor of the human Nav1.7 voltage gated sodium channel (IC50 = 28 nM). PF-04856264 blocks mouse Nav1.7 (IC50 = 131 nM) but has low potency against the rat Nav1.7 channel (IC50 = 4.2 mM).

Packaging

5, 25 mg in glass bottle

assay≥98% (HPLC)
colorwhite to light brown
formpowder
InChI keyMKSKJVIBSRUWSZ-UHFFFAOYSA-N
InChI1S/C20H15N5O3S2/c1-25-17(8-9-23-25)16-4-2-3-5-19(16)28-18-7-6-15(12-14(18)13-21)30(26,27)24-20-22-10-11-29-20/h2-12H,1H3,(H,22,24)
Quality Level100
SMILES stringO=S(C(C=C1)=CC(C#N)=C1OC2=CC=CC=C2C3=CC=NN3C)(NC4=NC=CS4)=O
solubilityDMSO: 10 mg/mL, clear
storage temp.2-8°C
Code
Description
Unit Size
List Price
Qty
SML1061-5MG
PF-04856264

Unit:5MG
List Price: £131.00
Source:List Price
ADD
Cas Number1235397-05-3
This product has met the following criteria: