SML0016-25MG Display Image

CCG-63802,

Code: SML0016-25MG D2-231

Application

CCG-63802 may be used to study G-protein-mediated cell signaling.

Biochem/physiol Actions

GCC-63802 binds to RGS4 and blocks interact...

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£320.30 25MG
List Price

Application

CCG-63802 may be used to study G-protein-mediated cell signaling.

Biochem/physiol Actions

GCC-63802 binds to RGS4 and blocks interaction with Goa (IC50 = 1.9 uM). RGS4 (Regulator of G protein Signaling) is one of the RGP proteins responsible for terminating mu opioid receptor signaling. RSG proteins are GTPase activators, and drive G protein subunits to an inactive, GDP-bound form.

Features and Benefits

This compound is featured on the G Proteins (Heterotrimeric) and Opioid Receptors pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

This compound is a featured product for Cyclic Nucleotide research. Click here to discover more featured Cyclic Nucleotide products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Packaging

5, 25 mg in glass bottle

storage temp.room temp
assay≥98% (HPLC)
solubilityDMSO: ≥5 mg/mL (;warmed DMSO)
Quality Level100
formpowder
coloryellow

Code
Description
Unit Size
List Price
Qty
SML0016-5MG
Unit:5MG
List Price: £85.59
Source:List Price
ADD
Cas Number0620112-78-9