E2661-5MG Display Image

Estropipate, >=98% (HPLC), powder

Code: E2661-5MG D2-231

Biochem/physiol Actions

Estropipate is the piperazine salt of the estrogen receptor agonist estrone-3-sulfate and a potent, specific inhibitor of the organic anion transporti...


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£136.00 5MG
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Biochem/physiol Actions

Estropipate is the piperazine salt of the estrogen receptor agonist estrone-3-sulfate and a potent, specific inhibitor of the organic anion transporting polypeptide 1B1 (OATP1B1, IC50 = 60 nM).

Features and Benefits

This compound is featured on the Nuclear Receptors (Steroids) page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

This compound was developed by Johnson & Johnson. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

This compound is a featured product for ADME Tox research. Click here to discover more featured ADME Tox products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Packaging

5, 25 mg in glass bottle

assay≥98% (HPLC)
colorwhite to tan
formpowder
Gene Informationhuman ... ESR1(2099)
InChI keyHZEQBCVBILBTEP-ZFINNJDLSA-N
InChI1S/C18H22O5S.C4H10N2/c1-18-9-8-14-13-5-3-12(23-24(20,21)22)10-11(13)2-4-15(14)16(18)6-7-17(18)19;1-2-6-4-3-5-1/h3,5,10,14-16H,2,4,6-9H2,1H3,(H,20,21,22);5-6H,1-4H2/t14-,15-,16+,18+;/m1./s1
optical activity[α]/D 100 to 120°, c = 1 in DMSO
originatorJohnson & Johnson
Quality Level100
SMILES stringC1CNCCN1.C[C@]23CC[C@H]4[C@@H](CCc5cc(OS(O)(=O)=O)ccc45)[C@@H]2CCC3=O
solubilityDMSO: ≥24 mg/mL
storage temp.2-8°C
Code
Description
Unit Size
List Price
Qty
E2661-25MG
Estropipate, >=98% (HPLC), powder

Unit:25MG
List Price: £376.00
Source:List Price
ADD
Cas Number7280-37-7
This product has met the following criteria: